PDB Information

PDB4MQU
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Small molecule disruptors of the glucokinase-glucokinase regulatory protein interaction: 2. Leveraging structure-based drug design to identify analogues with improved pharmacokinetic profiles.
St Jean, D.J., Ashton, K.S., Bartberger, M.D., Chen, J., Chmait, S., Cupples, R., Galbreath, E., Helmering, J., Hong, F.T., Jordan, S.R., Liu, L., Kunz, R.K., Michelsen, K., Nishimura, N., Pennington, L.D., Poon, S.F., Reid, D., Sivits, G., Stec, M.M., Tadesse, S., Tamayo, N., Van, G., Yang, K.C., Zhang, J., Norman, M.H., Fotsch, C., Lloyd, D.J., Hale, C.
J.Med.Chem.
HeaderTransferase Inhibitor
Released2013-09-16
Resolution2.220
CATH Insert Date11 May, 2014

PDB Images (9)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 12 May, 2014 Chopped
B 12 May, 2014 Chopped

CATH Domains (6)

Domain ID Date inserted into CATH Superfamily CATH Status
4mquA01 17 May, 2014 3.40.50.10490 Assigned
4mquA02 17 May, 2014 Holding pen
4mquA03 17 May, 2014 Holding pen
4mquB01 17 May, 2014 3.40.50.10490 Assigned
4mquB02 17 May, 2014 Holding pen
4mquB03 17 May, 2014 Holding pen

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q14397 GCKR_HUMAN Homo sapiens Glucokinase regulatory protein
Q14397 GCKR_HUMAN Homo sapiens Glucokinase regulatory protein