PDB Information

PDB4MPW
MethodX-RAY DIFFRACTION
Host OrganismKomagataella pastoris
Gene SourceHomo sapiens
Primary Citation
A Novel, Nonpeptidic, Orally Active Bivalent Inhibitor of Human beta-Tryptase.
Giardina, S.F., Werner, D.S., Pingle, M., Bergstrom, D.E., Arnold, L.D., Barany, F.
Pharmacology
HeaderHydrolase/Hydrolase Inhibitor
Released2013-09-13
Resolution1.950
CATH Insert Date28 Jun, 2015

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 29 Jun, 2015 Chopped
B 29 Jun, 2015 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
4mpwA01 09 Jul, 2015 2.40.10.10 Assigned
4mpwA02 09 Jul, 2015 2.40.10.10 Assigned
4mpwB01 10 Jul, 2015 2.40.10.10 Assigned
4mpwB02 10 Jul, 2015 2.40.10.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q15661 TRYB1_HUMAN Homo sapiens Tryptase alpha/beta-1
Q15661 TRYB1_HUMAN Homo sapiens Tryptase alpha/beta-1