PDB Information

PDB4MC9
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHuman immunodeficiency virus 1
Primary Citation
Structural Optimization of Cyclic Sulfonamide based Novel HIV-1 Protease Inhibitors to Pico Molar Affinities guided by X-ray Crystallographic Analysis
Ganguly, A.K., Alluri, S.S., Wang, C.H., Antropow, A., White, A., Caroccia, D., Biswas, D., Kang, E., Zhang, L.K., Carroll, S.S., Burlein, C., Fay, J., Orth, P., Strickland, C.
Tetrahedron
HeaderHydrolase/Hydrolase Inhibitor
Released2013-08-21
Resolution1.190
CATH Insert Date06 Apr, 2014

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 07 Apr, 2014 Chopped
B 07 Apr, 2014 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4mc9A00 25 Apr, 2014 2.40.70.10 Assigned
4mc9B00 25 Apr, 2014 2.40.70.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P0C6F2 POL_HV1LW Human immunodeficiency virus type 1 lw12.3 isolate Gag-Pol polyprotein
P0C6F2 POL_HV1LW Human immunodeficiency virus type 1 lw12.3 isolate Gag-Pol polyprotein