PDB Information

PDB4M3F
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceMycobacterium tuberculosis
Primary Citation
Ligand Efficiency Driven Design of New Inhibitors of Mycobacterium tuberculosis Transcriptional Repressor EthR Using Fragment Growing, Merging, and Linking Approaches.
Villemagne, B., Flipo, M., Blondiaux, N., Crauste, C., Malaquin, S., Leroux, F., Piveteau, C., Villeret, V., Brodin, P., Villoutreix, B.O., Sperandio, O., Soror, S.H., Wohlkonig, A., Wintjens, R., Deprez, B., Baulard, A.R., Willand, N.
J.Med.Chem.
HeaderTranscription Repressor/Inhibitor
Released2013-08-06
Resolution2.000
CATH Insert Date06 Jul, 2014

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 07 Jul, 2014 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4m3fA01 15 Jul, 2014 1.10.10.60 Assigned
4m3fA02 15 Jul, 2014 1.10.357.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P9WMC0 ETHR_MYCTO Mycobacterium tuberculosis CDC1551 HTH-type transcriptional regulator EthR