PDB 4l7f
PDB Information
| PDB | 4L7F |
| Method | X-RAY DIFFRACTION |
| Host Organism | |
| Gene Source | Homo sapiens |
| Primary Citation | Hit-to-lead optimization and kinase selectivity of imidazo[1,2-a]quinoxalin-4-amine derived JNK1 inhibitors.
Bioorg.Med.Chem.Lett.
|
| Header | Transferase/Transferase Inhibitor |
| Released | 2013-06-13 |
| Resolution | 1.950 |
| CATH Insert Date | 01 Sep, 2013 |
PDB Images (4)
PDB Prints
PDB Chains (1)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 02 Sep, 2013 | Chopped |
CATH Domains (2)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 4l7fA01 | 10 Sep, 2013 | 3.30.200.20 | Assigned |
| 4l7fA02 | 10 Sep, 2013 | 1.10.510.10 | Assigned |
UniProtKB Entries (1)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P45983 | MK08_HUMAN | Homo sapiens | Mitogen-activated protein kinase 8 |
