PDB 4kya
PDB Information
PDB | 4KYA |
Method | X-RAY DIFFRACTION |
Host Organism | Escherichia coli |
Gene Source | Toxoplasma gondii |
Primary Citation | Discovery of potent and selective inhibitors of Toxoplasma gondii thymidylate synthase for opportunistic infections.
ACS Med Chem Lett
|
Header | Oxidoreductase, Transferase/Inhibitor |
Released | 2013-05-28 |
Resolution | 3.260 |
CATH Insert Date | 24 Aug, 2014 |
PDB Images (33)
PDB Prints
PDB Chains (8)
Chain ID | Date inserted into CATH | CATH Status |
---|---|---|
A | 25 Aug, 2014 | Chopped |
B | 25 Aug, 2014 | Chopped |
C | 25 Aug, 2014 | Chopped |
D | 25 Aug, 2014 | Chopped |
E | 25 Aug, 2014 | Chopped |
F | 25 Aug, 2014 | Chopped |
G | 25 Aug, 2014 | Chopped |
H | 25 Aug, 2014 | Chopped |
CATH Domains (24)
Domain ID | Date inserted into CATH | Superfamily | CATH Status |
---|---|---|---|
4kyaA01 | 27 Aug, 2014 | 3.40.430.10 | Assigned |
4kyaA02 | 27 Aug, 2014 | Holding pen | |
4kyaA03 | 27 Aug, 2014 | 3.30.572.10 | Assigned |
4kyaB01 | 28 Aug, 2014 | 3.40.430.10 | Assigned |
4kyaB02 | 28 Aug, 2014 | Holding pen | |
4kyaB03 | 28 Aug, 2014 | 3.30.572.10 | Assigned |
4kyaC01 | 27 Aug, 2014 | 3.40.430.10 | Assigned |
4kyaC02 | 27 Aug, 2014 | Holding pen | |
4kyaC03 | 27 Aug, 2014 | 3.30.572.10 | Assigned |
4kyaD01 | 27 Aug, 2014 | 3.40.430.10 | Assigned |
4kyaD02 | 27 Aug, 2014 | Holding pen | |
4kyaD03 | 27 Aug, 2014 | 3.30.572.10 | Assigned |
4kyaE01 | 27 Aug, 2014 | 3.40.430.10 | Assigned |
4kyaE02 | 27 Aug, 2014 | Holding pen | |
4kyaE03 | 27 Aug, 2014 | 3.30.572.10 | Assigned |
4kyaF01 | 27 Aug, 2014 | 3.40.430.10 | Assigned |
4kyaF02 | 27 Aug, 2014 | Holding pen | |
4kyaF03 | 27 Aug, 2014 | 3.30.572.10 | Assigned |
4kyaG01 | 28 Aug, 2014 | 3.40.430.10 | Assigned |
4kyaG02 | 28 Aug, 2014 | Holding pen | |
4kyaG03 | 28 Aug, 2014 | 3.30.572.10 | Assigned |
4kyaH01 | 27 Aug, 2014 | 3.40.430.10 | Assigned |
4kyaH02 | 27 Aug, 2014 | Holding pen | |
4kyaH03 | 27 Aug, 2014 | 3.30.572.10 | Assigned |
UniProtKB Entries (8)
Accession | Gene ID | Taxon | Description |
---|---|---|---|
Q07422 | DRTS_TOXGO | Toxoplasma gondii | Bifunctional dihydrofolate reductase-thymidylate synthase |
Q07422 | DRTS_TOXGO | Toxoplasma gondii | Bifunctional dihydrofolate reductase-thymidylate synthase |
Q07422 | DRTS_TOXGO | Toxoplasma gondii | Bifunctional dihydrofolate reductase-thymidylate synthase |
Q07422 | DRTS_TOXGO | Toxoplasma gondii | Bifunctional dihydrofolate reductase-thymidylate synthase |
Q07422 | DRTS_TOXGO | Toxoplasma gondii | Bifunctional dihydrofolate reductase-thymidylate synthase |
Q07422 | DRTS_TOXGO | Toxoplasma gondii | Bifunctional dihydrofolate reductase-thymidylate synthase |
Q07422 | DRTS_TOXGO | Toxoplasma gondii | Bifunctional dihydrofolate reductase-thymidylate synthase |
Q07422 | DRTS_TOXGO | Toxoplasma gondii | Bifunctional dihydrofolate reductase-thymidylate synthase |