PDB Information

PDB4JT0
MethodX-RAY DIFFRACTION
Host Organism
Gene Source
Primary Citation
Dimerized Linear Mimics of a Natural Cyclopeptide (TMC-95A) Are Potent Noncovalent Inhibitors of the Eukaryotic 20S Proteasome
Desvergne, A., Genin, E., Marechal, X., Gallastegui, N., Dufau, L., Richy, N., Groll, M., Vidal, J., Reboud-Ravaux, M.
J.Med.Chem.
HeaderHydrolase/Hydrolase Inhibitor
Released2013-03-22
Resolution3.100
CATH Insert Date07 Jul, 2013

PDB Images (59)

PDB Prints

PDB Chains (30)

Chain ID Date inserted into CATH CATH Status
a 08 Jul, 2013 Chopped
A 08 Jul, 2013 Chopped
b 08 Jul, 2013 Chopped
B 08 Jul, 2013 Chopped
c 08 Jul, 2013 Rejected
C 08 Jul, 2013 Chopped
d 08 Jul, 2013 Rejected
D 08 Jul, 2013 Chopped
E 08 Jul, 2013 Chopped
F 08 Jul, 2013 Chopped
G 08 Jul, 2013 Chopped
H 08 Jul, 2013 Chopped
I 08 Jul, 2013 Chopped
J 08 Jul, 2013 Chopped
K 08 Jul, 2013 Chopped
L 08 Jul, 2013 Chopped
M 08 Jul, 2013 Chopped
N 08 Jul, 2013 Chopped
O 08 Jul, 2013 Chopped
P 08 Jul, 2013 Chopped
Q 08 Jul, 2013 Chopped
R 08 Jul, 2013 Chopped
S 08 Jul, 2013 Chopped
T 08 Jul, 2013 Chopped
U 08 Jul, 2013 Chopped
V 08 Jul, 2013 Chopped
W 08 Jul, 2013 Chopped
X 08 Jul, 2013 Chopped
Y 08 Jul, 2013 Chopped
Z 08 Jul, 2013 Chopped

CATH Domains (28)

Domain ID Date inserted into CATH Superfamily CATH Status
4jt0a00 09 Aug, 2013 3.60.20.10 Assigned
4jt0A00 09 Aug, 2013 3.60.20.10 Assigned
4jt0b00 09 Aug, 2013 3.60.20.10 Assigned
4jt0B00 09 Aug, 2013 3.60.20.10 Assigned
4jt0C00 09 Aug, 2013 3.60.20.10 Assigned
4jt0D00 09 Aug, 2013 3.60.20.10 Assigned
4jt0E00 09 Aug, 2013 3.60.20.10 Assigned
4jt0F00 09 Aug, 2013 3.60.20.10 Assigned
4jt0G00 09 Aug, 2013 3.60.20.10 Assigned
4jt0H00 09 Aug, 2013 3.60.20.10 Assigned
4jt0I00 09 Aug, 2013 3.60.20.10 Assigned
4jt0J00 09 Aug, 2013 3.60.20.10 Assigned
4jt0K00 09 Aug, 2013 3.60.20.10 Assigned
4jt0L00 09 Aug, 2013 3.60.20.10 Assigned
4jt0M00 09 Aug, 2013 3.60.20.10 Assigned
4jt0N00 09 Aug, 2013 3.60.20.10 Assigned
4jt0O00 09 Aug, 2013 3.60.20.10 Assigned
4jt0P00 09 Aug, 2013 3.60.20.10 Assigned
4jt0Q00 09 Aug, 2013 3.60.20.10 Assigned
4jt0R00 09 Aug, 2013 3.60.20.10 Assigned
4jt0S00 09 Aug, 2013 3.60.20.10 Assigned
4jt0T00 09 Aug, 2013 3.60.20.10 Assigned
4jt0U00 09 Aug, 2013 3.60.20.10 Assigned
4jt0V00 09 Aug, 2013 3.60.20.10 Assigned
4jt0W00 09 Aug, 2013 3.60.20.10 Assigned
4jt0X00 09 Aug, 2013 3.60.20.10 Assigned
4jt0Y00 09 Aug, 2013 3.60.20.10 Assigned
4jt0Z00 09 Aug, 2013 3.60.20.10 Assigned

UniProtKB Entries (28)

Accession Gene ID Taxon Description
P40302 PSA6_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-6
P21242 PSA7_YEAST Saccharomyces cerevisiae S288C Probable proteasome subunit alpha type-7
P38624 PSB1_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-1
P32379 PSA5_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-5
P40303 PSA4_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-4
P23638 PSA3_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-3
P23639 PSA2_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-2
P23724 PSB6_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-6
P23724 PSB6_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-6
P21243 PSA1_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-1
P30657 PSB7_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-7
P21242 PSA7_YEAST Saccharomyces cerevisiae S288C Probable proteasome subunit alpha type-7
P40303 PSA4_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-4
P30657 PSB7_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-7
P23638 PSA3_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-3
P40302 PSA6_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-6
P25451 PSB3_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-3
P21243 PSA1_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-1
P30656 PSB5_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-5
P23639 PSA2_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-2
P25043 PSB2_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-2
P25451 PSB3_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-3
P22141 PSB4_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-4
P22141 PSB4_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-4
P38624 PSB1_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-1
P25043 PSB2_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-2
P30656 PSB5_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-5
P32379 PSA5_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-5