PDB Information

PDB4J5P
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceRattus norvegicus
Primary Citation
Rational design of Fatty Acid amide hydrolase inhibitors that act by covalently bonding to two active site residues.
Otrubova, K., Brown, M., McCormick, M.S., Han, G.W., O'Neal, S.T., Cravatt, B.F., Stevens, R.C., Lichtman, A.H., Boger, D.L.
J.Am.Chem.Soc.
HeaderHydrolase/Hydrolase Inhibitor
Released2013-02-08
Resolution2.300
CATH Insert Date07 Jul, 2013

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 08 Jul, 2013 Chopped
B 08 Jul, 2013 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4j5pA00 09 Aug, 2013 3.90.1300.10 Assigned
4j5pB00 09 Aug, 2013 3.90.1300.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P97612 FAAH1_RAT Rattus norvegicus Fatty-acid amide hydrolase 1
P97612 FAAH1_RAT Rattus norvegicus Fatty-acid amide hydrolase 1