PDB Information

PDB4IU6
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Pyridinylquinazolines selectively inhibit human methionine aminopeptidase-1 in cells.
Zhang, F., Bhat, S., Gabelli, S.B., Chen, X., Miller, M.S., Nacev, B.A., Cheng, Y.L., Meyers, D.J., Tenney, K., Shim, J.S., Crews, P., Amzel, L.M., Ma, D., Liu, J.O.
J.Med.Chem.
HeaderHydrolase/Hydrolase Inhibitor
Released2013-01-19
Resolution1.900
CATH Insert Date07 Jul, 2013

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 08 Jul, 2013 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
4iu6A00 13 Sep, 2013 3.90.230.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P53582 MAP11_HUMAN Homo sapiens Methionine aminopeptidase 1