PDB Information

PDB4IKF
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHuman spumaretrovirus
Primary Citation
2-Hydroxyisoquinoline-1,3(2H,4H)-diones (HIDs), novel inhibitors of HIV integrase with a high barrier to resistance.
Desimmie, B.A., Demeulemeester, J., Suchaud, V., Taltynov, O., Billamboz, M., Lion, C., Bailly, F., Strelkov, S.V., Debyser, Z., Cotelle, P., Christ, F.
Acs Chem.Biol.
HeaderViral Protein/Dna/Inhibitor
Released2012-12-26
Resolution3.400
CATH Insert Date07 Jul, 2013

PDB Images (10)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 08 Jul, 2013 Chopped
B 08 Jul, 2013 Chopped
C 08 Jul, 2013 Rejected
D 08 Jul, 2013 Rejected

CATH Domains (5)

Domain ID Date inserted into CATH Superfamily CATH Status
4ikfA01 30 Aug, 2013 1.10.340.70 Assigned
4ikfA02 30 Aug, 2013 2.30.30.140 Assigned
4ikfA03 30 Aug, 2013 3.30.420.10 Assigned
4ikfA04 30 Aug, 2013 6.10.20.110 Assigned
4ikfB00 09 Aug, 2013 3.30.420.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P14350 POL_FOAMV Human spumaretrovirus Pro-Pol polyprotein
P14350 POL_FOAMV Human spumaretrovirus Pro-Pol polyprotein