PDB Information

PDB4IEH
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
The role of the acidity of N-heteroaryl sulfonamides as inhibitors of bcl-2 family protein-protein interactions.
Toure, B.B., Miller-Moslin, K., Yusuff, N., Perez, L., Dore, M., Joud, C., Michael, W., DiPietro, L., van der Plas, S., McEwan, M., Lenoir, F., Hoe, M., Karki, R., Springer, C., Sullivan, J., Levine, K., Fiorilla, C., Xie, X., Kulathila, R., Herlihy, K., Porter, D., Visser, M.
ACS Med Chem Lett
HeaderApoptosis/Inhibitor
Released2012-12-13
Resolution2.100
CATH Insert Date04 Aug, 2013

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 05 Aug, 2013 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
4iehA00 28 Aug, 2013 Holding pen

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P10415 BCL2_HUMAN Homo sapiens Apoptosis regulator Bcl-2
Q07817 B2CL1_HUMAN Homo sapiens Bcl-2-like protein 1