PDB Information

PDB4I9Z
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Exploration of the 5-bromopyrimidin-4(3H)-ones as potent inhibitors of PDE5.
Gong, X., Wang, G., Ren, J., Liu, Z., Wang, Z., Chen, T., Yang, X., Jiang, X., Shen, J., Jiang, H., Aisa, H.A., Xu, Y., Li, J.
Bioorg.Med.Chem.Lett.
HeaderHydrolase/Hydrolase Inhibitor
Released2012-12-05
Resolution2.080
CATH Insert Date05 Jan, 2014

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 06 Jan, 2014 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
4i9zA00 09 Jan, 2014 1.10.1300.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
O76074 PDE5A_HUMAN Homo sapiens cGMP-specific 3',5'-cyclic phosphodiesterase