PDB Information

PDB4I4E
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Structure-based discovery of cellular-active allosteric inhibitors of FAK.
Tomita, N., Hayashi, Y., Suzuki, S., Oomori, Y., Aramaki, Y., Matsushita, Y., Iwatani, M., Iwata, H., Okabe, A., Awazu, Y., Isono, O., Skene, R.J., Hosfield, D.J., Miki, H., Kawamoto, T., Hori, A., Baba, A.
Bioorg.Med.Chem.Lett.
HeaderTransferase/Transferase Inhibitor
Released2012-11-27
Resolution1.550
CATH Insert Date28 Mar, 2013

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 28 Mar, 2013 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4i4eA01 14 Aug, 2013 3.30.200.20 Assigned
4i4eA02 14 Aug, 2013 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
Q05397 FAK1_HUMAN Homo sapiens Focal adhesion kinase 1