PDB 4i41
PDB Information
| PDB | 4I41 |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli |
| Gene Source | Homo sapiens |
| Primary Citation | A new target for an old drug: identifying mitoxantrone as a nanomolar inhibitor of PIM1 kinase via kinome-wide selectivity modeling.
J. Med. Chem.
|
| Header | Transferase/Transferase Inhibitor |
| Released | 2012-11-27 |
| Resolution | 2.700 |
| CATH Insert Date | 15 Dec, 2013 |
PDB Images (4)
PDB Prints
PDB Chains (1)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 16 Dec, 2013 | Chopped |
CATH Domains (2)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 4i41A01 | 20 Dec, 2013 | 3.30.200.20 | Assigned |
| 4i41A02 | 20 Dec, 2013 | 1.10.510.10 | Assigned |
UniProtKB Entries (1)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P11309 | PIM1_HUMAN | Homo sapiens | Serine/threonine-protein kinase pim-1 |
