PDB Information

PDB4HVS
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Design and pharmacology of a highly specific dual FMS and KIT kinase inhibitor.
Zhang, C., Ibrahim, P.N., Zhang, J., Burton, E.A., Habets, G., Zhang, Y., Powell, B., West, B.L., Matusow, B., Tsang, G., Shellooe, R., Carias, H., Nguyen, H., Marimuthu, A., Zhang, K.Y., Oh, A., Bremer, R., Hurt, C.R., Artis, D.R., Wu, G., Nespi, M., Spevak, W., Lin, P., Nolop, K., Hirth, P., Tesch, G.H., Bollag, G.
Proc.Natl.Acad.Sci.USA
HeaderTransferase/Transferase Inhibitor
Released2012-11-06
Resolution1.900
CATH Insert Date07 Jul, 2013

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 08 Jul, 2013 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4hvsA01 09 Aug, 2013 3.30.200.20 Assigned
4hvsA02 09 Aug, 2013 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P10721 KIT_HUMAN Homo sapiens Mast/stem cell growth factor receptor Kit