PDB 4hvb
PDB Information
| PDB | 4HVB |
| Method | X-RAY DIFFRACTION |
| Host Organism | Spodoptera frugiperda |
| Gene Source | Homo sapiens |
| Primary Citation | Discovery of the Highly Potent PI3K/mTOR Dual Inhibitor PF-04979064 through Structure-Based Drug Design.
ACS Med Chem Lett
|
| Header | Transferase/Transferase Inhibitor |
| Released | 2012-11-05 |
| Resolution | 2.350 |
| CATH Insert Date | 24 Nov, 2013 |
PDB Images (7)
PDB Prints
PDB Chains (1)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 25 Nov, 2013 | Chopped |
CATH Domains (5)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 4hvbA01 | 27 Nov, 2013 | 3.10.20.90 | Assigned |
| 4hvbA02 | 27 Nov, 2013 | 2.60.40.150 | Assigned |
| 4hvbA03 | 27 Nov, 2013 | 1.25.40.70 | Assigned |
| 4hvbA04 | 27 Nov, 2013 | 3.30.1010.10 | Assigned |
| 4hvbA05 | 27 Nov, 2013 | 1.10.1070.11 | Assigned |
UniProtKB Entries (1)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P48736 | PK3CG_HUMAN | Homo sapiens | Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform |
