PDB Information

PDB4HRC
MethodX-RAY DIFFRACTION
Host Organism
Gene Source
Primary Citation
Enzyme inhibition by hydroamination: design and mechanism of a hybrid carmaphycin-syringolin enone proteasome inhibitor.
Trivella, D.B., Pereira, A.R., Stein, M.L., Kasai, Y., Byrum, T., Valeriote, F.A., Tantillo, D.J., Groll, M., Gerwick, W.H., Moore, B.S.
Chem.Biol.
HeaderHydrolase/Hydrolase Inhibitor
Released2012-10-27
Resolution2.800
CATH Insert Date02 Feb, 2014

PDB Images (57)

PDB Prints

PDB Chains (28)

Chain ID Date inserted into CATH CATH Status
a 03 Feb, 2014 Chopped
A 03 Feb, 2014 Chopped
b 03 Feb, 2014 Chopped
B 03 Feb, 2014 Chopped
C 03 Feb, 2014 Chopped
D 03 Feb, 2014 Chopped
E 03 Feb, 2014 Chopped
F 03 Feb, 2014 Chopped
G 03 Feb, 2014 Chopped
H 03 Feb, 2014 Chopped
I 03 Feb, 2014 Chopped
J 03 Feb, 2014 Chopped
K 03 Feb, 2014 Chopped
L 03 Feb, 2014 Chopped
M 03 Feb, 2014 Chopped
N 03 Feb, 2014 Chopped
O 03 Feb, 2014 Chopped
P 03 Feb, 2014 Chopped
Q 03 Feb, 2014 Chopped
R 03 Feb, 2014 Chopped
S 03 Feb, 2014 Chopped
T 03 Feb, 2014 Chopped
U 03 Feb, 2014 Chopped
V 03 Feb, 2014 Chopped
W 03 Feb, 2014 Chopped
X 03 Feb, 2014 Chopped
Y 03 Feb, 2014 Chopped
Z 03 Feb, 2014 Chopped

CATH Domains (28)

Domain ID Date inserted into CATH Superfamily CATH Status
4hrca00 07 Mar, 2014 3.60.20.10 Assigned
4hrcA00 07 Mar, 2014 3.60.20.10 Assigned
4hrcb00 07 Mar, 2014 3.60.20.10 Assigned
4hrcB00 07 Mar, 2014 3.60.20.10 Assigned
4hrcC00 07 Mar, 2014 3.60.20.10 Assigned
4hrcD00 07 Mar, 2014 3.60.20.10 Assigned
4hrcE00 07 Mar, 2014 3.60.20.10 Assigned
4hrcF00 07 Mar, 2014 3.60.20.10 Assigned
4hrcG00 07 Mar, 2014 3.60.20.10 Assigned
4hrcH00 07 Mar, 2014 3.60.20.10 Assigned
4hrcI00 07 Mar, 2014 3.60.20.10 Assigned
4hrcJ00 07 Mar, 2014 3.60.20.10 Assigned
4hrcK00 07 Mar, 2014 3.60.20.10 Assigned
4hrcL00 07 Mar, 2014 3.60.20.10 Assigned
4hrcM00 07 Mar, 2014 3.60.20.10 Assigned
4hrcN00 07 Mar, 2014 3.60.20.10 Assigned
4hrcO00 07 Mar, 2014 3.60.20.10 Assigned
4hrcP00 07 Mar, 2014 3.60.20.10 Assigned
4hrcQ00 07 Mar, 2014 3.60.20.10 Assigned
4hrcR00 07 Mar, 2014 3.60.20.10 Assigned
4hrcS00 07 Mar, 2014 3.60.20.10 Assigned
4hrcT00 07 Mar, 2014 3.60.20.10 Assigned
4hrcU00 07 Mar, 2014 3.60.20.10 Assigned
4hrcV00 07 Mar, 2014 3.60.20.10 Assigned
4hrcW00 07 Mar, 2014 3.60.20.10 Assigned
4hrcX00 07 Mar, 2014 3.60.20.10 Assigned
4hrcY00 07 Mar, 2014 3.60.20.10 Assigned
4hrcZ00 07 Mar, 2014 3.60.20.10 Assigned

UniProtKB Entries (28)

Accession Gene ID Taxon Description
P40303 PSA4_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-4
P25043 PSB2_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-2
P21243 PSA1_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-1
P30657 PSB7_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-7
P21242 PSA7_YEAST Saccharomyces cerevisiae S288C Probable proteasome subunit alpha type-7
P23639 PSA2_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-2
P40302 PSA6_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-6
P21242 PSA7_YEAST Saccharomyces cerevisiae S288C Probable proteasome subunit alpha type-7
P38624 PSB1_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-1
P23639 PSA2_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-2
P25451 PSB3_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-3
P25043 PSB2_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-2
P23638 PSA3_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-3
P23638 PSA3_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-3
P23724 PSB6_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-6
P38624 PSB1_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-1
P40303 PSA4_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-4
P25451 PSB3_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-3
P22141 PSB4_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-4
P30656 PSB5_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-5
P32379 PSA5_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-5
P40302 PSA6_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-6
P23724 PSB6_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-6
P21243 PSA1_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-1
P30657 PSB7_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-7
P22141 PSB4_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-4
P30656 PSB5_YEAST Saccharomyces cerevisiae S288C Proteasome subunit beta type-5
P32379 PSA5_YEAST Saccharomyces cerevisiae S288C Proteasome subunit alpha type-5