PDB 4hee
PDB Information
| PDB | 4HEE |
| Method | X-RAY DIFFRACTION |
| Host Organism | Spodoptera frugiperda |
| Gene Source | Homo sapiens |
| Primary Citation | Design, synthesis, and evaluation of imidazo[4,5-c]pyridin-4-one derivatives with dual activity at angiotensin II type 1 receptor and peroxisome proliferator-activated receptor-gamma
Bioorg.Med.Chem.Lett.
|
| Header | Transcription/Transcription Inhibitor |
| Released | 2012-10-03 |
| Resolution | 2.500 |
| CATH Insert Date | 01 Sep, 2013 |
PDB Images (4)
PDB Prints
PDB Chains (2)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| X | 02 Sep, 2013 | Chopped |
| Y | 02 Sep, 2013 | Rejected |
CATH Domains (1)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 4heeX00 | 10 Sep, 2013 | 1.10.565.10 | Assigned |
UniProtKB Entries (2)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| Q15788 | NCOA1_HUMAN | Homo sapiens | Nuclear receptor coactivator 1 |
| P37231 | PPARG_HUMAN | Homo sapiens | Peroxisome proliferator-activated receptor gamma |
