PDB 4gpj

PDB Information

PDB4GPJ
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
The design and synthesis of 5- and 6-isoxazolylbenzimidazoles as selective inhibitors of the BET Bromodomains
Hay, D., Fedorov, O., Filippakopoulos, P., Picaud, S., Martin, S., Philpott, M., Hewings, D., Uttakar, S., Heightman, T.D., Conway, S., Knapp, S., Brennan, P.
TO BE PUBLISHED
HeaderProtein Binding/Inhibitor
Released2012-08-21
Resolution1.600
CATH Insert Date04 Nov, 2012

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 05 Nov, 2012 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
4gpjA01 10 Nov, 2012 1.20.920.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
O60885 BRD4_HUMAN Homo sapiens Bromodomain-containing protein 4
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