PDB 4geb
PDB Information
| PDB | 4GEB |
| Method | X-RAY DIFFRACTION |
| Host Organism | Spodoptera frugiperda |
| Gene Source | Homo sapiens |
| Primary Citation | PF-04859989 as a template for structure-based drug design: identification of new pyrazole series of irreversible KAT II inhibitors with improved lipophilic efficiency.
Bioorg.Med.Chem.Lett.
|
| Header | Transferase/Transferase Inhibitor |
| Released | 2012-08-01 |
| Resolution | 2.150 |
| CATH Insert Date | 28 Mar, 2013 |
PDB Images (9)
PDB Prints
PDB Chains (2)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 28 Mar, 2013 | Chopped |
| B | 28 Mar, 2013 | Chopped |
CATH Domains (6)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 4gebA01 | 30 Aug, 2013 | Holding pen | |
| 4gebA02 | 30 Aug, 2013 | 3.40.640.10 | Assigned |
| 4gebA03 | 30 Aug, 2013 | 3.90.1150.10 | Assigned |
| 4gebB01 | 30 Aug, 2013 | Holding pen | |
| 4gebB02 | 30 Aug, 2013 | 3.40.640.10 | Assigned |
| 4gebB03 | 30 Aug, 2013 | 3.90.1150.10 | Assigned |
UniProtKB Entries (2)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| Q8N5Z0 | AADAT_HUMAN | Homo sapiens | Kynurenine/alpha-aminoadipate aminotransferase, mitochondrial |
| Q8N5Z0 | AADAT_HUMAN | Homo sapiens | Kynurenine/alpha-aminoadipate aminotransferase, mitochondrial |
