PDB Information

PDB4G8R
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Mechanistic characterization and crystal structure of a small molecule inactivator bound to plasminogen activator inhibitor-1.
Li, S.H., Reinke, A.A., Sanders, K.L., Emal, C.D., Whisstock, J.C., Stuckey, J.A., Lawrence, D.A.
Proc.Natl.Acad.Sci.USA
HeaderBlood Clotting/Inhibitor
Released2012-07-23
Resolution2.190
CATH Insert Date05 Jan, 2014

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 06 Jan, 2014 Chopped
B 06 Jan, 2014 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
4g8rA01 09 Jan, 2014 3.30.497.10 Assigned
4g8rA02 09 Jan, 2014 2.30.39.10 Assigned
4g8rB01 09 Jan, 2014 3.30.497.10 Assigned
4g8rB02 09 Jan, 2014 2.30.39.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P05121 PAI1_HUMAN Homo sapiens Plasminogen activator inhibitor 1
P05121 PAI1_HUMAN Homo sapiens Plasminogen activator inhibitor 1