PDB Information

PDB4G2F
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Discovery of a novel chemotype of tyrosine kinase inhibitors by fragment-based docking and molecular dynamics.
Zhao, H., Dong, J., Lafleur, K., Nevado, C., Caflisch, A.
ACS MED.CHEM.LETT.
HeaderTransferase/Transferase Inhibitor
Released2012-07-12
Resolution1.700
CATH Insert Date04 Nov, 2012

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 05 Nov, 2012 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4g2fA01 10 Nov, 2012 3.30.200.20 Assigned
4g2fA02 10 Nov, 2012 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P29320 EPHA3_HUMAN Homo sapiens Ephrin type-A receptor 3