PDB Information

PDB4FCF
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceKlebsiella pneumoniae
Primary Citation
Design and exploration of novel boronic acid inhibitors reveals important interactions with a clavulanic acid-resistant sulfhydryl-variable (SHV) beta-lactamase.
Winkler, M.L., Rodkey, E.A., Taracila, M.A., Drawz, S.M., Bethel, C.R., Papp-Wallace, K.M., Smith, K.M., Xu, Y., Dwulit-Smith, J.R., Romagnoli, C., Caselli, E., Prati, F., van den Akker, F., Bonomo, R.A.
J.Med.Chem.
HeaderHydrolase/Hydrolase Inhibitor
Released2012-05-24
Resolution1.090
CATH Insert Date30 Dec, 2012

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 31 Dec, 2012 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
4fcfA00 08 Feb, 2013 3.40.710.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P0AD64 BLA1_KLEPN Klebsiella pneumoniae Beta-lactamase SHV-1