PDB 4e90
PDB Information
PDB | 4E90 |
Method | X-RAY DIFFRACTION |
Host Organism | |
Gene Source | Homo sapiens |
Primary Citation | Application of structure-based drug design and parallel chemistry to identify selective, brain penetrant, in vivo active phosphodiesterase 9A inhibitors.
J.Med.Chem.
|
Header | Hydrolase/Hydrolase Inhibitor |
Released | 2012-03-20 |
Resolution | 2.500 |
CATH Insert Date | 28 Mar, 2013 |
PDB Images (5)
PDB Prints
PDB Chains (2)
Chain ID | Date inserted into CATH | CATH Status |
---|---|---|
A | 28 Mar, 2013 | Chopped |
B | 28 Mar, 2013 | Chopped |
CATH Domains (2)
Domain ID | Date inserted into CATH | Superfamily | CATH Status |
---|---|---|---|
4e90A00 | 10 Apr, 2013 | 1.10.1300.10 | Assigned |
4e90B00 | 10 Apr, 2013 | 1.10.1300.10 | Assigned |
UniProtKB Entries (2)
Accession | Gene ID | Taxon | Description |
---|---|---|---|
O76083 | PDE9A_HUMAN | Homo sapiens | High affinity cGMP-specific 3',5'-cyclic phosphodiesterase 9A |
O76083 | PDE9A_HUMAN | Homo sapiens | High affinity cGMP-specific 3',5'-cyclic phosphodiesterase 9A |