PDB Information

PDB4E7R
MethodX-RAY DIFFRACTION
Host Organism
Gene Source
Primary Citation
New 3-amidinophenylalanine-derived inhibitors of matriptase
Hammami, M., Ruehmann, E., Mauerer, M., Heine, A., Guetschow, M., Klebe, G., Steinmetzer, T.
MEDCHEMCOMM
HeaderHydrolase/Hydrolase Inhibitor
Released2012-03-19
Resolution2.250
CATH Insert Date24 Jun, 2012

PDB Images (11)

PDB Prints

PDB Chains (6)

Chain ID Date inserted into CATH CATH Status
G 24 Jun, 2012 Chopped
H 24 Jun, 2012 Chopped
I 24 Jun, 2012 Rejected
J 24 Jun, 2012 Rejected
L 24 Jun, 2012 Rejected
M 24 Jun, 2012 Rejected

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
4e7rG01 28 Jun, 2012 2.40.10.10 Assigned
4e7rG02 28 Jun, 2012 2.40.10.10 Assigned
4e7rH01 28 Jun, 2012 2.40.10.10 Assigned
4e7rH02 28 Jun, 2012 2.40.10.10 Assigned

UniProtKB Entries (6)

Accession Gene ID Taxon Description
P00734 THRB_HUMAN Homo sapiens Prothrombin
P09945 HIRV2_HIRME Hirudo medicinalis Hirudin variant-2
P09945 HIRV2_HIRME Hirudo medicinalis Hirudin variant-2
P00734 THRB_HUMAN Homo sapiens Prothrombin
P00734 THRB_HUMAN Homo sapiens Prothrombin
P00734 THRB_HUMAN Homo sapiens Prothrombin