PDB Information

PDB4CDE
MethodX-RAY DIFFRACTION
Host OrganismSPODOPTERA FRUGIPERDA
Gene SourceHOMO SAPIENS
Primary Citation
Cathepsin C Inhibitors: Property Optimization and Identification of a Clinical Candidate.
Furber, M., Gardiner, P., Tiden, A.K., Mete, A., Ford, R., Millichip, I., Stein, L., Mather, A., Kinchin, E., Luckhurst, C., Barber, S., Cage, P., Sanganee, H., Austin, R., Chohan, K., Beri, R., Thong, B., Wallace, A., Oreffo, V., Hutchinson, R., Harper, S., Debreczeni, J., Breed, J., Wissler, L., Edman, K.
J.Med.Chem.
HeaderHydrolase
Released2013-10-31
Resolution2.400
CATH Insert Date23 Mar, 2014

PDB Images (13)

PDB Prints

PDB Chains (6)

Chain ID Date inserted into CATH CATH Status
A 24 Mar, 2014 Chopped
B 24 Mar, 2014 Chopped
C 24 Mar, 2014 Chopped
D 24 Mar, 2014 Chopped
E 24 Mar, 2014 Chopped
F 24 Mar, 2014 Chopped

CATH Domains (6)

Domain ID Date inserted into CATH Superfamily CATH Status
4cdeA00 25 Apr, 2014 2.40.128.80 Assigned
4cdeB01 25 Apr, 2014 3.90.70.10 Assigned
4cdeC00 25 Apr, 2014 2.40.50.170 Assigned
4cdeD00 25 Apr, 2014 2.40.128.80 Assigned
4cdeE01 17 Apr, 2014 3.90.70.10 Assigned
4cdeF00 25 Apr, 2014 2.40.50.170 Assigned

UniProtKB Entries (6)

Accession Gene ID Taxon Description
P53634 CATC_HUMAN Homo sapiens Dipeptidyl peptidase 1
P53634 CATC_HUMAN Homo sapiens Dipeptidyl peptidase 1
P53634 CATC_HUMAN Homo sapiens Dipeptidyl peptidase 1
P53634 CATC_HUMAN Homo sapiens Dipeptidyl peptidase 1
P53634 CATC_HUMAN Homo sapiens Dipeptidyl peptidase 1
P53634 CATC_HUMAN Homo sapiens Dipeptidyl peptidase 1