PDB Information

PDB4BGH
MethodX-RAY DIFFRACTION
Host OrganismSPODOPTERA FRUGIPERDA
Gene SourceHOMO SAPIENS
Primary Citation
The Lab Oddity Prevails: Discovery of Pan-Cdk Inhibitor (R)- S-Cyclopropyl-S-(4-{[4-{[(1R,2R)-2-Hydroxy-1-Methylpropyl]Oxy}-5-(Trifluoromethyl)Pyrimidin-2-Yl]Amino}Phenyl)Sulfoximide (Bay 1000394) for the Treatment of Cancer.
Lucking, U., Jautelat, R., Kruger, M., Brumby, T., Lienau, P., Schafer, M., Briem, H., Schulze, J., Hillisch, A., Reichel, A., Wengner, A.M., Siemeister, G.
Chemmedchem
HeaderTransferase
Released2013-03-26
Resolution1.950
CATH Insert Date22 Sep, 2013

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 23 Sep, 2013 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4bghA01 25 Sep, 2013 3.30.200.20 Assigned
4bghA02 25 Sep, 2013 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P24941 CDK2_HUMAN Homo sapiens Cyclin-dependent kinase 2