PDB Information

PDB4A9R
MethodX-RAY DIFFRACTION
Host OrganismESCHERICHIA COLI
Gene SourceHOMO SAPIENS
Primary Citation
Benzimidazole Inhibitors of the Protein Kinase Chk2: Clarification of the Binding Mode by Flexible Side Chain Docking and Protein-Ligand Crystallography
Matijssen, C., Silva-Santisteban, M.C., Westwood, I.M., Siddique, S., Choi, V., Sheldrake, P., Van Montfort, R.L.M., Blagg, J.
Bioorg.Med.Chem.
HeaderTransferase
Released2011-11-28
Resolution2.850
CATH Insert Date04 Nov, 2012

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 05 Nov, 2012 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4a9rA01 18 Apr, 2013 3.30.200.20 Assigned
4a9rA02 18 Apr, 2013 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
O96017 CHK2_HUMAN Homo sapiens Serine/threonine-protein kinase Chk2