PDB Information

PDB4A33
MethodX-RAY DIFFRACTION
Host OrganismESCHERICHIA COLI
Gene SourceLEISHMANIA MAJOR
Primary Citation
Discovery of a novel class of orally active trypanocidal N-myristoyltransferase inhibitors.
Brand, S., Cleghorn, L.A., McElroy, S.P., Robinson, D.A., Smith, V.C., Hallyburton, I., Harrison, J.R., Norcross, N.R., Spinks, D., Bayliss, T., Norval, S., Stojanovski, L., Torrie, L.S., Frearson, J.A., Brenk, R., Fairlamb, A.H., Ferguson, M.A., Read, K.D., Wyatt, P.G., Gilbert, I.H.
J. Med. Chem.
HeaderTransferase
Released2011-09-29
Resolution2.400
CATH Insert Date08 Jan, 2012

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 09 Jan, 2012 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
4a33A00 28 Aug, 2013 3.40.630.170 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
Q4Q5S8 Q4Q5S8_LEIMA Leishmania major Glycylpeptide N-tetradecanoyltransferase