PDB 3zim
PDB Information
| PDB | 3ZIM |
| Method | X-RAY DIFFRACTION |
| Host Organism | SPODOPTERA FRUGIPERDA |
| Gene Source | HOMO SAPIENS |
| Primary Citation | Discovery of a Potent and Isoform-Selective Targeted Covalent Inhibitor of the Lipid Kinase Pi3Kalpha
J.Med.Chem.
|
| Header | Transferase |
| Released | 2013-01-09 |
| Resolution | 2.850 |
| CATH Insert Date | 28 Mar, 2013 |
PDB Images (7)
PDB Prints
PDB Chains (1)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 28 Mar, 2013 | Chopped |
CATH Domains (5)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 3zimA01 | 21 Nov, 2013 | 3.10.20.90 | Assigned |
| 3zimA02 | 21 Nov, 2013 | 2.60.40.150 | Assigned |
| 3zimA03 | 21 Nov, 2013 | 1.25.40.70 | Assigned |
| 3zimA04 | 21 Nov, 2013 | 3.30.1010.10 | Assigned |
| 3zimA05 | 21 Nov, 2013 | 1.10.1070.11 | Assigned |
UniProtKB Entries (1)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P42336 | PK3CA_HUMAN | Homo sapiens | Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform |
