PDB 3wzj

PDB Information

PDB3WZJ
MethodX-RAY DIFFRACTION
Host OrganismCELL-FREE SYNTHESIS
Gene SourceHomo sapiens
Primary Citation
Discovery of Imidazo[1,2-b]pyridazine Derivatives: Selective and Orally Available Mps1 (TTK) Kinase Inhibitors Exhibiting Remarkable Antiproliferative Activity
Kusakabe, K.I., Ide, N., Daigo, Y., Itoh, T., Yamamoto, T., Hashizume, H., Nozu, K., Yoshida, H., Tadano, G., Tagashira, S., Higashino, K., Okano, Y., Sato, Y., Inoue, M., Iguchi, M., Kanazawa, T., Ishioka, Y., Dohi, K., Kido, Y., Sakamoto, S., Ando, S., Maeda, M., Higaki, M., Baba, Y., Nakamura, Y.
J.Med.Chem.
HeaderTransferase
Released2014-09-29
Resolution2.750
CATH Insert Date28 Jun, 2015

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 29 Jun, 2015 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
3wzjA01 10 Jul, 2015 3.30.200.20 Assigned
3wzjA02 10 Jul, 2015 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P33981 TTK_HUMAN Homo sapiens Dual specificity protein kinase TTK