PDB Information

PDB3WAX
MethodX-RAY DIFFRACTION
Host OrganismHomo Sapiens
Gene SourceMus musculus
Primary Citation
Screening and X-ray Crystal Structure-based Optimization of Autotaxin (ENPP2) Inhibitors, Using a Newly Developed Fluorescence Probe
Kawaguchi, M., Okabe, T., Okudaira, S., Nishimasu, H., Ishitani, R., Kojima, H., Nureki, O., Aoki, J., Nagano, T.
Acs Chem.Biol.
HeaderHydrolase/Hydrolase Inhibitor
Released2013-05-09
Resolution1.900
CATH Insert Date18 Aug, 2013

PDB Images (6)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 19 Aug, 2013 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
3waxA01 04 Nov, 2013 4.10.410.20 Assigned
3waxA02 04 Nov, 2013 4.10.410.20 Assigned
3waxA03 04 Nov, 2013 3.40.720.10 Assigned
3waxA04 04 Nov, 2013 3.40.570.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
Q9R1E6 ENPP2_MOUSE Mus musculus Ectonucleotide pyrophosphatase/phosphodiesterase family member 2