PDB 3u5k
PDB Information
| PDB | 3U5K |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli |
| Gene Source | Homo sapiens |
| Primary Citation | Benzodiazepines and benzotriazepines as protein interaction inhibitors targeting bromodomains of the BET family.
Bioorg.Med.Chem.
|
| Header | Signaling Protein/Inhibitor |
| Released | 2011-10-11 |
| Resolution | 1.800 |
| CATH Insert Date | 27 Nov, 2011 |
PDB Images (9)
PDB Prints
PDB Chains (4)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 29 Nov, 2011 | Chopped |
| B | 29 Nov, 2011 | Chopped |
| C | 29 Nov, 2011 | Chopped |
| D | 29 Nov, 2011 | Chopped |
CATH Domains (4)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 3u5kA01 | 01 Dec, 2011 | 1.20.920.10 | Assigned |
| 3u5kB01 | 01 Dec, 2011 | 1.20.920.10 | Assigned |
| 3u5kC01 | 01 Dec, 2011 | 1.20.920.10 | Assigned |
| 3u5kD01 | 01 Dec, 2011 | 1.20.920.10 | Assigned |
UniProtKB Entries (4)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| O60885 | BRD4_HUMAN | Homo sapiens | Bromodomain-containing protein 4 |
| O60885 | BRD4_HUMAN | Homo sapiens | Bromodomain-containing protein 4 |
| O60885 | BRD4_HUMAN | Homo sapiens | Bromodomain-containing protein 4 |
| O60885 | BRD4_HUMAN | Homo sapiens | Bromodomain-containing protein 4 |
