PDB 3t9i
PDB Information
| PDB | 3T9I |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli |
| Gene Source | Homo sapiens |
| Primary Citation | Discovery of novel 3,5-disubstituted indole derivatives as potent inhibitors of Pim-1, Pim-2, and Pim-3 protein kinases.
Bioorg.Med.Chem.Lett.
|
| Header | Transferase/Transferase Inhibitor |
| Released | 2011-08-02 |
| Resolution | 2.600 |
| CATH Insert Date | 16 Oct, 2011 |
PDB Images (4)
PDB Prints
PDB Chains (1)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 29 Nov, 2011 | Chopped |
CATH Domains (2)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 3t9iA01 | 01 Dec, 2011 | 3.30.200.20 | Assigned |
| 3t9iA02 | 01 Dec, 2011 | 1.10.510.10 | Assigned |
UniProtKB Entries (1)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P11309 | PIM1_HUMAN | Homo sapiens | Serine/threonine-protein kinase pim-1 |
