PDB Information

PDB3SR4
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Selective Inhibitors of Histone Methyltransferase DOT1L: Design, Synthesis, and Crystallographic Studies.
Yao, Y., Chen, P., Diao, J., Cheng, G., Deng, L., Anglin, J.L., Prasad, B.V., Song, Y.
J.Am.Chem.Soc.
HeaderTransferase/Transferase Inhibitor
Released2011-07-06
Resolution2.500
CATH Insert Date09 Oct, 2011

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 29 Nov, 2011 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
3sr4A01 01 Dec, 2011 1.10.260.60 Assigned
3sr4A02 01 Dec, 2011 3.40.50.150 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
Q8TEK3 DOT1L_HUMAN Homo sapiens Histone-lysine N-methyltransferase, H3 lysine-79 specific