PDB Information

PDB3SHE
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Novel ATP competitive MK2 inhibitors with potent biochemical and cell-based activity throughout the series.
Oubrie, A., Kaptein, A., de Zwart, E., Hoogenboom, N., Goorden, R., van de Kar, B., van Hoek, M., de Kimpe, V., van der Heijden, R., Borsboom, J., Kazemier, B., de Roos, J., Scheffers, M., Lommerse, J., Schultz-Fademrecht, C., Barf, T.
Bioorg.Med.Chem.Lett.
HeaderTransferase/Transferase Inhibitor
Released2011-06-16
Resolution2.250
CATH Insert Date08 Jan, 2012

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 09 Jan, 2012 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
3sheA01 16 Jan, 2012 3.30.200.20 Assigned
3sheA02 16 Jan, 2012 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
Q16644 MAPK3_HUMAN Homo sapiens MAP kinase-activated protein kinase 3