PDB Information

PDB3R0T
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Unprecedented selectivity and structural determinants of a new class of protein kinase CK2 inhibitors in clinical trials for the treatment of cancer.
Battistutta, R., Cozza, G., Pierre, F., Papinutto, E., Lolli, G., Sarno, S., O'Brien, S.E., Siddiqui-Jain, A., Haddach, M., Anderes, K., Ryckman, D.M., Meggio, F., Pinna, L.A.
Biochemistry
HeaderTransferase/Transferase Inhibitor
Released2011-03-09
Resolution1.750
CATH Insert Date11 Dec, 2011

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 12 Dec, 2011 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
3r0tA01 16 Jan, 2012 1.10.510.10 Assigned
3r0tA02 16 Jan, 2012 3.30.200.20 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P68400 CSK21_HUMAN Homo sapiens Casein kinase II subunit alpha