PDB Information

PDB3QTI
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
A Drug Resistance Screen Using a Selective MET Inhibitor Reveals a Spectrum of Mutations That Partially Overlap with Activating Mutations Found in Cancer Patients.
Tiedt, R., Degenkolbe, E., Furet, P., Appleton, B.A., Wagner, S., Schoepfer, J., Buck, E., Ruddy, D.A., Monahan, J.E., Jones, M.D., Blank, J., Haasen, D., Drueckes, P., Wartmann, M., McCarthy, C., Sellers, W.R., Hofmann, F.
Cancer Res.
HeaderTransferase/Transferase Inhibitor
Released2011-02-22
Resolution2.000
CATH Insert Date24 Jul, 2011

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 01 Aug, 2011 Chopped
B 01 Aug, 2011 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
3qtiA01 12 Aug, 2011 3.30.200.20 Assigned
3qtiA02 12 Aug, 2011 1.10.510.10 Assigned
3qtiB01 12 Aug, 2011 3.30.200.20 Assigned
3qtiB02 12 Aug, 2011 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P08581 MET_HUMAN Homo sapiens Hepatocyte growth factor receptor
P08581 MET_HUMAN Homo sapiens Hepatocyte growth factor receptor