Discovery and Optimization of a Series of Benzothiazole Phosphoinositide 3-Kinase (PI3K)/Mammalian Target of Rapamycin (mTOR) Dual Inhibitors.
D'Angelo, N.D., Kim, T.S., Andrews, K., Booker, S.K., Caenepeel, S., Chen, K., D'Amico, D., Freeman, D., Jiang, J., Liu, L., McCarter, J.D., San Miguel, T., Mullady, E.L., Schrag, M., Subramanian, R., Tang, J., Wahl, R.C., Wang, L., Whittington, D.A., Wu, T., Xi, N., Xu, Y., Yakowec, P., Yang, K., Zalameda, L.P., Zhang, N., Hughes, P., Norman, M.H.
J.Med.Chem.