PDB Information

PDB3Q0V
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceMycobacterium tuberculosis
Primary Citation
Design, synthesis and optimization of new EthR inhibitors. A new alternative approach to fight tuberculosis by boosting ethionamide
Flipo, M., Desroses, M., Dirie, B., Carette, X., Leroux, F., Lens, Z., Rucktooa, P., Leroux, F., Piveteau, C., Demirkaya, F., Locht, C., Villeret, V., Christophe, T., Jeon, H.K., Brodin, P., Deprez, B., Baulard, A., Willand, N.
To be Published
HeaderTranscription/Transcription Inhibitor
Released2010-12-16
Resolution1.950
CATH Insert Date15 Jan, 2012

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 16 Jan, 2012 Chopped
B 16 Jan, 2012 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
3q0vA01 19 Jan, 2012 1.10.10.60 Assigned
3q0vA02 19 Jan, 2012 1.10.357.10 Assigned
3q0vB01 19 Jan, 2012 1.10.10.60 Assigned
3q0vB02 19 Jan, 2012 1.10.357.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P9WMC1 ETHR_MYCTU Mycobacterium tuberculosis H37Rv HTH-type transcriptional regulator EthR
P9WMC1 ETHR_MYCTU Mycobacterium tuberculosis H37Rv HTH-type transcriptional regulator EthR