PDB 3p88

PDB Information

PDB3P88
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Conformationally constrained farnesoid X receptor (FXR) agonists: Heteroaryl replacements of the naphthalene.
Bass, J.Y., Caravella, J.A., Chen, L., Creech, K.L., Deaton, D.N., Madauss, K.P., Marr, H.B., McFadyen, R.B., Miller, A.B., Mills, W.Y., Navas, F., Parks, D.J., Smalley, T.L., Spearing, P.K., Todd, D., Williams, S.P., Wisely, G.B.
Bioorg.Med.Chem.Lett.
HeaderTranscription/Inhibitor
Released2010-10-13
Resolution2.950
CATH Insert Date04 Sep, 2011

PDB Images (4)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 05 Sep, 2011 Chopped
B 05 Sep, 2011 Rejected

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
3p88A00 06 Sep, 2011 1.10.565.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q15788 NCOA1_HUMAN Homo sapiens Nuclear receptor coactivator 1
Q96RI1 NR1H4_HUMAN Homo sapiens Bile acid receptor