PDB Information

PDB3OY3
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceMus musculus
Primary Citation
Structural Mechanism of the Pan-BCR-ABL Inhibitor Ponatinib (AP24534): Lessons for Overcoming Kinase Inhibitor Resistance.
Zhou, T., Commodore, L., Huang, W.S., Wang, Y., Thomas, M., Keats, J., Xu, Q., Rivera, V.M., Shakespeare, W.C., Clackson, T., Dalgarno, D.C., Zhu, X.
Chem.Biol.Drug Des.
HeaderTransferase/Transferase Inhibitor
Released2010-09-22
Resolution1.950
CATH Insert Date23 Jan, 2011

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 24 Jan, 2011 Chopped
B 24 Jan, 2011 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
3oy3A01 17 Feb, 2011 3.30.200.20 Assigned
3oy3A02 17 Feb, 2011 1.10.510.10 Assigned
3oy3B01 17 Feb, 2011 3.30.200.20 Assigned
3oy3B02 17 Feb, 2011 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P00520 ABL1_MOUSE Mus musculus Tyrosine-protein kinase ABL1
P00520 ABL1_MOUSE Mus musculus Tyrosine-protein kinase ABL1