PDB Information

PDB3NW6
MethodX-RAY DIFFRACTION
Host Organismunidentified BACULOVIRUS
Gene SourceHomo sapiens
Primary Citation
Proline isosteres in a series of 2,4-disubstituted pyrrolo[1,2-f][1,2,4]triazine inhibitors of IGF-1R kinase and IR kinase.
Sampognaro, A.J., Wittman, M.D., Carboni, J.M., Chang, C., Greer, A.F., Hurlburt, W.W., Sack, J.S., Vyas, D.M.
Bioorg.Med.Chem.Lett.
HeaderTransferase
Released2010-07-09
Resolution2.200
CATH Insert Date15 Aug, 2010

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 16 Aug, 2010 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
3nw6A01 17 Feb, 2011 3.30.200.20 Assigned
3nw6A02 17 Feb, 2011 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P08069 IGF1R_HUMAN Homo sapiens Insulin-like growth factor 1 receptor