PDB Information

PDB3MVJ
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Design of selective, ATP-competitive inhibitors of Akt.
Freeman-Cook, K.D., Autry, C., Borzillo, G., Gordon, D., Barbacci-Tobin, E., Bernardo, V., Briere, D., Clark, T., Corbett, M., Jakubczak, J., Kakar, S., Knauth, E., Lippa, B., Luzzio, M.J., Mansour, M., Martinelli, G., Marx, M., Nelson, K., Pandit, J., Rajamohan, F., Robinson, S., Subramanyam, C., Wei, L., Wythes, M., Morris, J.
J.Med.Chem.
HeaderTransferase
Released2010-05-04
Resolution2.490
CATH Insert Date06 Jun, 2010

PDB Images (13)

PDB Prints

PDB Chains (6)

Chain ID Date inserted into CATH CATH Status
A 06 Jun, 2010 Chopped
B 06 Jun, 2010 Chopped
E 06 Jun, 2010 Chopped
I 06 Jun, 2010 Rejected
J 06 Jun, 2010 Rejected
K 06 Jun, 2010 Rejected

CATH Domains (6)

Domain ID Date inserted into CATH Superfamily CATH Status
3mvjA01 03 Aug, 2010 1.10.510.10 Assigned
3mvjA02 03 Aug, 2010 3.30.200.20 Assigned
3mvjB01 03 Aug, 2010 1.10.510.10 Assigned
3mvjB02 03 Aug, 2010 3.30.200.20 Assigned
3mvjE01 03 Aug, 2010 1.10.510.10 Assigned
3mvjE02 03 Aug, 2010 3.30.200.20 Assigned

UniProtKB Entries (3)

Accession Gene ID Taxon Description
P17612 KAPCA_HUMAN Homo sapiens cAMP-dependent protein kinase catalytic subunit alpha
P17612 KAPCA_HUMAN Homo sapiens cAMP-dependent protein kinase catalytic subunit alpha
P17612 KAPCA_HUMAN Homo sapiens cAMP-dependent protein kinase catalytic subunit alpha