PDB 3mjw
PDB Information
| PDB | 3MJW |
| Method | X-RAY DIFFRACTION |
| Host Organism | Spodoptera frugiperda |
| Gene Source | Homo sapiens |
| Primary Citation | 5-Ureidobenzofuranone indoles as potent and efficacious inhibitors of PI3 kinase-alpha and mTOR for the treatment of breast cancer.
Bioorg.Med.Chem.Lett.
|
| Header | Transferase |
| Released | 2010-04-13 |
| Resolution | 2.870 |
| CATH Insert Date | 13 Jun, 2010 |
PDB Images (7)
PDB Prints
PDB Chains (1)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 13 Jun, 2010 | Chopped |
CATH Domains (5)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 3mjwA01 | 31 Jul, 2010 | 3.10.20.90 | Assigned |
| 3mjwA02 | 31 Jul, 2010 | 2.60.40.150 | Assigned |
| 3mjwA03 | 31 Jul, 2010 | 1.25.40.70 | Assigned |
| 3mjwA04 | 31 Jul, 2010 | 3.30.1010.10 | Assigned |
| 3mjwA05 | 31 Jul, 2010 | 1.10.1070.11 | Assigned |
UniProtKB Entries (1)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P48736 | PK3CG_HUMAN | Homo sapiens | Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform |
