PDB Information

PDB3KWJ
MethodX-RAY DIFFRACTION
Host OrganismPichia pastoris
Gene SourceHomo sapiens
Primary Citation
Aryl- and heteroaryl-substituted aminobenzo[a]quinolizines as dipeptidyl peptidase IV inhibitors.
Boehringer, M., Fischer, H., Hennig, M., Hunziker, D., Huwyler, J., Kuhn, B., Loeffler, B.M., Luebbers, T., Mattei, P., Narquizian, R., Sebokova, E., Sprecher, U., Wessel, H.P.
Bioorg.Med.Chem.Lett.
HeaderHydrolase
Released2009-12-01
Resolution2.800
CATH Insert Date19 Sep, 2010

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 20 Sep, 2010 Chopped
B 20 Sep, 2010 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
3kwjA01 26 Sep, 2010 3.40.50.1820 Assigned
3kwjA02 26 Sep, 2010 2.140.10.30 Assigned
3kwjB01 27 Sep, 2010 3.40.50.1820 Assigned
3kwjB02 27 Sep, 2010 2.140.10.30 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P27487 DPP4_HUMAN Homo sapiens Dipeptidyl peptidase 4
P27487 DPP4_HUMAN Homo sapiens Dipeptidyl peptidase 4