PDB Information

PDB3KSQ
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceRattus norvegicus
Primary Citation
Discovery of C-imidazole azaheptapyridine FPT inhibitors.
Zhu, H.Y., Cooper, A.B., Desai, J., Njoroge, G., Kirschmeier, P., Bishop, W.R., Strickland, C., Hruza, A., Doll, R.J., Girijavallabhan, V.M.
Bioorg.Med.Chem.Lett.
HeaderTransferase
Released2009-11-23
Resolution2.100
CATH Insert Date31 Jan, 2010

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 31 Jan, 2010 Chopped
B 31 Jan, 2010 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
3ksqA00 27 Jun, 2010 1.25.40.120 Assigned
3ksqB00 27 Jun, 2010 1.50.10.20 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q04631 FNTA_RAT Rattus norvegicus Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha
Q02293 FNTB_RAT Rattus norvegicus Protein farnesyltransferase subunit beta