PDB Information

PDB3KL6
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Discovery of a tetrahydropyrimidin-2(1H)-one derivative (TAK-442) as a potent, selective, and orally active factor Xa inhibitor.
Fujimoto, T., Imaeda, Y., Konishi, N., Hiroe, K., Kawamura, M., Textor, G.P., Aertgeerts, K., Kubo, K.
J.Med.Chem.
HeaderHydrolase
Released2009-11-06
Resolution1.450
CATH Insert Date03 Dec, 2009

PDB Images (6)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 03 Dec, 2009 Chopped
B 03 Dec, 2009 Chopped

CATH Domains (3)

Domain ID Date inserted into CATH Superfamily CATH Status
3kl6A01 19 Apr, 2010 2.40.10.10 Assigned
3kl6A02 19 Apr, 2010 2.40.10.10 Assigned
3kl6B00 19 Apr, 2010 2.10.25.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P00742 FA10_HUMAN Homo sapiens Coagulation factor X
P00742 FA10_HUMAN Homo sapiens Coagulation factor X