PDB Information

PDB3KFC
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
4-(3-Aryloxyaryl)quinoline sulfones are potent liver X receptor agonists.
Bernotas, R.C., Singhaus, R.R., Kaufman, D.H., Travins, J.M., Ullrich, J.W., Unwalla, R., Quinet, E., Evans, M., Nambi, P., Olland, A., Kauppi, B., Wilhelmsson, A., Goos-Nilsson, A., Wrobel, J.
Bioorg.Med.Chem.Lett.
HeaderTranscription
Released2009-10-27
Resolution2.400
CATH Insert Date10 Dec, 2009

PDB Images (9)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 10 Dec, 2009 Chopped
B 10 Dec, 2009 Chopped
C 10 Dec, 2009 Chopped
D 10 Dec, 2009 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
3kfcA00 04 Feb, 2013 1.10.565.10 Assigned
3kfcB00 04 Feb, 2013 1.10.565.10 Assigned
3kfcC00 16 Apr, 2010 1.10.565.10 Assigned
3kfcD00 04 Feb, 2013 1.10.565.10 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
P55055 NR1H2_HUMAN Homo sapiens Oxysterols receptor LXR-beta
P55055 NR1H2_HUMAN Homo sapiens Oxysterols receptor LXR-beta
P55055 NR1H2_HUMAN Homo sapiens Oxysterols receptor LXR-beta
P55055 NR1H2_HUMAN Homo sapiens Oxysterols receptor LXR-beta