PDB 3kc0
PDB Information
| PDB | 3KC0 |
| Method | X-RAY DIFFRACTION |
| Host Organism | Escherichia coli |
| Gene Source | Homo sapiens |
| Primary Citation | Structure-based drug design of tricyclic 8H-indeno[1,2-d][1,3]thiazoles as potent FBPase inhibitors.
Bioorg.Med.Chem.Lett.
|
| Header | Hydrolase |
| Released | 2009-10-20 |
| Resolution | 2.800 |
| CATH Insert Date | 07 Feb, 2010 |
PDB Images (13)
PDB Prints
PDB Chains (4)
| Chain ID | Date inserted into CATH | CATH Status |
|---|---|---|
| A | 08 Feb, 2010 | Chopped |
| B | 08 Feb, 2010 | Chopped |
| C | 08 Feb, 2010 | Chopped |
| D | 08 Feb, 2010 | Chopped |
CATH Domains (8)
| Domain ID | Date inserted into CATH | Superfamily | CATH Status |
|---|---|---|---|
| 3kc0A01 | 15 Apr, 2010 | 3.30.540.10 | Assigned |
| 3kc0A02 | 15 Apr, 2010 | 3.40.190.80 | Assigned |
| 3kc0B01 | 15 Apr, 2010 | 3.30.540.10 | Assigned |
| 3kc0B02 | 15 Apr, 2010 | 3.40.190.80 | Assigned |
| 3kc0C01 | 15 Apr, 2010 | 3.30.540.10 | Assigned |
| 3kc0C02 | 15 Apr, 2010 | 3.40.190.80 | Assigned |
| 3kc0D01 | 15 Apr, 2010 | 3.30.540.10 | Assigned |
| 3kc0D02 | 15 Apr, 2010 | 3.40.190.80 | Assigned |
UniProtKB Entries (4)
| Accession | Gene ID | Taxon | Description |
|---|---|---|---|
| P09467 | F16P1_HUMAN | Homo sapiens | Fructose-1,6-bisphosphatase 1 |
| P09467 | F16P1_HUMAN | Homo sapiens | Fructose-1,6-bisphosphatase 1 |
| P09467 | F16P1_HUMAN | Homo sapiens | Fructose-1,6-bisphosphatase 1 |
| P09467 | F16P1_HUMAN | Homo sapiens | Fructose-1,6-bisphosphatase 1 |
